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Home - Products - Endocrinology/Hormones - Opioid Receptor - (±)-U-50488 hydrochloride

(±)-U-50488 hydrochloride

CAS No. 67197-96-0

(±)-U-50488 hydrochloride( U50488 | U-50488 )

Catalog No. M15564 CAS No. 67197-96-0

A potent, selective kappa-opioid receptor agonist with no μ-opioid antagonist effects.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    (±)-U-50488 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective kappa-opioid receptor agonist with no μ-opioid antagonist effects.
  • Description
    A potent, selective kappa-opioid receptor agonist with no μ-opioid antagonist effects; shows analgesic, diuretic and antitussive effects, and reverses the memory impairment produced by anticholinergic drugs in vivo.Anxiety Discontinued.
  • In Vitro
    (±)-U-50488 is a racemic mixture of (+)-Trans-(1R,2R)-U-50488 and (-)-Trans-(1S,2S)-U-50488.
  • In Vivo
    ——
  • Synonyms
    U50488 | U-50488
  • Pathway
    Endocrinology/Hormones
  • Target
    Opioid Receptor
  • Recptor
    Opioid Receptor
  • Research Area
    Neurological Disease
  • Indication
    Anxiety

Chemical Information

  • CAS Number
    67197-96-0
  • Formula Weight
    405.79
  • Molecular Formula
    C19H26Cl2N2O.HCl
  • Purity
    >98% (HPLC)
  • Solubility
    25 mM in H2O
  • SMILES
    CN(C1CCCCC1N2CCCC2)C(=O)CC3=CC(=C(C=C3)Cl)Cl.CN(C1CCCCC1N2CCCC2)C(=O)CC3=CC(=C(C=C3)Cl)Cl.Cl.Cl
  • Chemical Name
    trans-(±)-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]benzeneacetamide hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Tao PL, et al. Eur J Pharmacol. 1994 May 2;256(3):281-6. 2. Suarez-Roca H, et al. J Pharmacol Exp Ther. 1993 Feb;264(2):648-53. 3. Su MT, et al. Br J Pharmacol. 1998 Feb;123(4):625-30. 4. Vonvoigtlander PF, et al. J Pharmacol Exp Ther. 1983 Jan;224(1):7-12.
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